Our current publications
These are current publications by researchers at the Department of Medicinal Chemistry. You can always contact us for more information on our results.
Part of Biochimica et Biophysica Acta - Biomembranes, 2024
Article in journal
- DOI for A closer look at calcium-induced interactions between phosphatidylserine-(PS) doped liposomes and the structural effects caused by inclusion of gangliosides or polyethylene glycol- (PEG) modified lipids
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A film-like SERS aptasensor for sensitive detection of patulin based on GO@Au nanosheets
Part of Food Chemistry, 2024
Article in journal
A small-angle X-ray scattering study of amphiphilic drug self-assemblies in polyacrylate microgels
Part of Colloids and Surfaces A, 2024
Article in journal
- DOI for A small-angle X-ray scattering study of amphiphilic drug self-assemblies in polyacrylate microgels
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Part of Pharmaceuticals, 2024
Article in journal
- DOI for Advancements in Microfluidic Cassette-Based iMiDEVTM Technology for Production of L-[11C]Methionine and [11C]Choline
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Part of Acta neuropathologica communications, 2024
Article in journal
- DOI for Altered amyloid-β structure markedly reduces gliosis in the brain of mice harboring the Uppsala APP deletion
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Part of Clinical Microbiology and Infection, p. 256-257, 2024
Article in journal
Atypical Complications during the Course of COVID-19: A Comprehensive Review
Part of Medicina, 2024
Article, review/survey
- DOI for Atypical Complications during the Course of COVID-19: A Comprehensive Review
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Part of Food Chemistry, 2024
Article in journal
Part of Molecular Pharmaceutics, p. 1919-1932, 2024
Article in journal
Part of EJNMMI Radiopharmacy and Chemistry, 2024
Article in journal
- DOI for Comparison of approaches for increasing affinity of affibody molecules for imaging of B7-H3: dimerization and affinity maturation
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Part of PLOS ONE, 2024
Article in journal
- DOI for Comparison of EKFC, Pakistani CKD-EPI and 2021 Race-Free CKD-EPI creatinine equations in South Asian CKD population: A study from Pakistani CKD community cohort
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Engineering and characterization of a hydrogel mimicking subcutaneous interstitial space
Part of European Polymer Journal, 2024
Article in journal
- DOI for Engineering and characterization of a hydrogel mimicking subcutaneous interstitial space
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Enhanced Risk Assessment of Transformation Products through Chemical Similarity Analysis
Part of ACS - ES & T Water, p. 1949-1951, 2024
Article in journal
- DOI for Enhanced Risk Assessment of Transformation Products through Chemical Similarity Analysis
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Part of BMC Infectious Diseases, 2024
Article in journal
- DOI for Evaluation of clinical and laboratory characteristics of dengue viral infection and risk factors of dengue hemorrhagic fever: a multi-center retrospective analysis
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Formulation and evaluation of miconazole lipogel for enhanced drug permeation
Part of Pakistan Journal of Pharmaceutical Sciences, p. 95-105, 2024
Article in journal
Part of Pharmaceutics, 2024
Article in journal
- DOI for GRPR-Antagonists Carrying DOTAGA-Chelator via Positively Charged Linkers: Perspectives for Prostate Cancer Theranostics
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Part of Journal of Controlled Release, p. 468-478, 2024
Article in journal
- DOI for Half-life extension via ABD-fusion leads to higher tumor uptake of an affibody-drug conjugate compared to PAS- and XTENylation.
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Identification of New Ketamine Metabolites and Their Detailed Distribution in the Mammalian Brain
Part of ACS Chemical Neuroscience, p. 1335-1341, 2024
Article in journal
- DOI for Identification of New Ketamine Metabolites and Their Detailed Distribution in the Mammalian Brain
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Part of International Journal of Molecular Sciences, 2024
Article in journal
- DOI for Influence of Molecular Design on the Tumor Targeting and Biodistribution of PSMA-Binding Tracers Labeled with Technetium-99m
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Part of Molecular Metabolism, 2024
Article in journal
- DOI for Inhibiting the endoplasmic reticulum stress response enhances the effect of doxorubicin by altering the lipid metabolism of liver cancer cells
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Inhibition of Insulin-Regulated Aminopeptidase by Imidazo[1,5-α]pyridines; Synthesis and Evaluation
Part of International Journal of Molecular Sciences, 2024
Article in journal
- DOI for Inhibition of Insulin-Regulated Aminopeptidase by Imidazo[1,5-α]pyridines; Synthesis and Evaluation
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Part of Nuclear Medicine and Biology, 2024
Article in journal
- DOI for Introduction of a fatty acid chain modification to prolong circulatory half-life of a radioligand towards glucose-dependent insulinotropic polypeptide receptor
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Part of Soft Matter, p. 2272-2279, 2024
Article in journal
- DOI for Investigation of supramolecular structures in various aqueous solutions of an amyloid forming peptide using small-angle X-ray scattering
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Part of Physical Chemistry, Chemical Physics - PCCP, 2024
Article in journal
N-(Heteroaryl)thiophene sulfonamides as angiotensin AT2 receptor ligands
Part of European Journal of Medicinal Chemistry, 2024
Article in journal
- DOI for N-(Heteroaryl)thiophene sulfonamides as angiotensin AT2 receptor ligands
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Part of Journal of Agricultural and Food Chemistry, p. 9691-9702, 2024
Article in journal
Preclinical Evaluation of HER2-Targeting DARPin G3: Impact of Albumin-Binding Domain (ABD) Fusion
Part of International Journal of Molecular Sciences, 2024
Article in journal
- DOI for Preclinical Evaluation of HER2-Targeting DARPin G3: Impact of Albumin-Binding Domain (ABD) Fusion
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Part of EJNMMI Radiopharmacy and Chemistry, 2024
Article in journal
- DOI for Preclinical evaluation of new GRPR-antagonists with improved metabolic stability for radiotheranostic use in oncology
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Part of ACS Omega, p. 10522-10538, 2024
Article in journal
- DOI for Preparation and Evaluation of a Self-Emulsifying Drug Delivery System for Improving the Solubility and Permeability of Ticagrelor
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Part of Environmental Science and Technology, p. 7078-7086, 2024
Article in journal
- DOI for Preparation of Simple Bicyclic Carboxylate-Rich Alicyclic Molecules for the Investigation of Dissolved Organic Matter
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Part of Molecular Medicine Reports, 2024
Article in journal
- DOI for Reduction of renal activity retention of radiolabeled albumin binding domain-derived affinity proteins using a non-residualizing label strategy compared with a cleavable glycine-leucine-glycine-lysine-linker
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Part of Saudi Pharmaceutical Journal, 2024
Article in journal
- DOI for Response Surface Methodology (RSM) approach to formulate and optimize the bilayer combination tablet of Tamsulosin and Finasteride
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Part of PLOS ONE, 2024
Article in journal
- DOI for Screening for antibacterial and cytotoxic activities of Sri Lankan marine sponges through microfractionation: Isolation of bromopyrrole alkaloids from Stylissa massa
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Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
Part of EJNMMI Radiopharmacy and Chemistry, 2024
Article in journal
- DOI for Synthesis and evaluation of fluorine-18 labelled tetrazines as pre-targeting imaging agents for PET
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Part of ACS Pharmacology & Translational Science, p. 1457-1473, 2024
Article in journal
Part of Hormones and Behavior, 2024
Article in journal
- DOI for The decanoate esters of nandrolone, testosterone, and trenbolone induce steroid specific memory impairment and somatic effects in the male rat
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Part of International Journal of Molecular Sciences, 2024
Article in journal
- DOI for The Discovery of New Inhibitors of Insulin-Regulated Aminopeptidase by a High-Throughput Screening of 400,000 Drug-like Compounds
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Part of FOOD SCIENCE AND HUMAN WELLNESS, p. 146-153, 2024
Article in journal
- DOI for Three novel umami peptides derived from the alcohol extract of the Pacific oyster (Crassostrea gigas): identification, characterizations and interactions with T1R1/T1R3 taste receptors
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Part of ACS Omega, p. 18608-18616, 2024
Article in journal
- DOI for Two Novel [68Ga]Ga-Labeled Radiotracers Based on Metabolically Stable [Sar11]RM26 Antagonistic Peptide for Diagnostic Positron Emission Tomography Imaging of GRPR-Positive Prostate Cancer
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Part of Peptides, 2024
Article in journal
- DOI for Venomous gland transcriptome and venom proteomic analysis of the scorpion Androctonus amoreuxi reveal new peptides with anti-SARS-CoV-2 activity
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Part of Frontiers in Oncology, 2023
Article in journal
- DOI for 177Lu-labeled PSMA targeting therapeutic with optimized linker for treatment of disseminated prostate cancer; evaluation of biodistribution and dosimetry
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[18F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44
Part of Pharmaceutics, 2023
Article in journal
- DOI for [18F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44
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A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane
Part of Advanced Synthesis and Catalysis, p. 1839-1845, 2023
Article in journal
- DOI for A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane
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Part of Journal of chromatography. B, 2023
Article in journal
- DOI for A multivariate data analysis approach for the investigation of in vitro derived metabolites of ACP-105 in comparison with human in vivo metabolites
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Part of Comprehensive Psychiatry, 2023
Article in journal
- DOI for Acute nicotine exposure blocks aromatase in the limbic brain of healthy women: A [11C]cetrozole PET study
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Acyl Amidines by Pd-Catalyzed Aminocarbonylation: One-Pot Cyclizations and C-11 Labeling
Part of Journal of Organic Chemistry, p. 5078-5089, 2023
Article in journal
- DOI for Acyl Amidines by Pd-Catalyzed Aminocarbonylation: One-Pot Cyclizations and C-11 Labeling
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Part of Electrophoresis, p. 1247-1257, 2023
Article in journal
- DOI for An interlaboratory capillary zone electrophoresis-UV study of various monoclonal antibodies, instruments, and ε-aminocaproic acid lots
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An overview of surface forces and the DLVO theory
Part of ChemTexts, 2023
Article in journal
- DOI for An overview of surface forces and the DLVO theory
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Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents
Part of ACS Medicinal Chemistry Letters, p. 802-809, 2023
Article in journal
Part of International Journal of Polymer Science, 2023
Article in journal
- DOI for Application of Nanoprecipitation Technique to Develop Poloxamer-407 Facilitated Solid Lipid Nanoparticles for the Controlled Delivery of Tacrolimus
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